Publicação

Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control

Ver documento

Detalhes bibliográficos
Resumo:Additive manufacturing advancements contribute considerably to several fields, and its use in the medical field is gaining attention due to its easily customizable option (patient-specific), low cost, and fast turnout time in developing drug delivery and diagnostic tools. Here, wereport the fabrication of a microneedle (MN) platform using a stereolithography 3D printer, varying the 3D printing angle and aspect ratio (2:1, 3:1, 4:1). The optimal printing angle was30, resulting in needle tip and base diameters of 50 µm and 330 µm, and heights of 550/850/1180 µm. Polyvinyl alcohol (PVA) MNs produced with varying levofloxacin concentrations showed variability of 4% in tip and 3% base diameters and 15% in height compared to the 3D-printed MNs. Geometry B wasused to produce levofloxacin-loaded PVA MNs and tested against Klebsiella pneumoniae colony biofilms. Levofloxacin wasreleased gradually, as assessed by spectrofluorimetry. The MIC of levofloxacin against the K. pneumoniae clinical isolate was4 µg/mL, but this concentration wasinsufficient to cause any effect on K. pneumoniae biofilms. Only concentrations 32 µg/mL werestatistically different compared to the unloaded MNs. 3D printing is an attractive solution to produce molds for fabricating biopolymeric MNs for topical drug delivery.
Autores principais:Vinayakumar, K. B.
Outros Autores:Silva, Maria Daniela; Martins, Artur; Mundy, Stephen; González-Losada, Pedro; Sillankorva, Sanna M.
Assunto:3D printing biofilms Klebsiella pneumoniae levofloxacin microneedles polyvinyl alcohol
Ano:2023
País:Portugal
Tipo de documento:artigo
Tipo de acesso:acesso aberto
Instituição associada:Universidade do Minho
Idioma:inglês
Origem:RepositóriUM - Universidade do Minho
_version_ 1867438274680717312
author Vinayakumar, K. B.
author2 Silva, Maria Daniela
Martins, Artur
Mundy, Stephen
González-Losada, Pedro
Sillankorva, Sanna M.
author2_role author
author
author
author
author
author_facet Vinayakumar, K. B.
Silva, Maria Daniela
Martins, Artur
Mundy, Stephen
González-Losada, Pedro
Sillankorva, Sanna M.
author_role author
contributor_name_str_mv RepositóriUM - Universidade do Minho
country_str PT
creators_json_txt [{\"Person.name\":\"Vinayakumar, K. B.\"},{\"Person.name\":\"Silva, Maria Daniela\"},{\"Person.name\":\"Martins, Artur\"},{\"Person.name\":\"Mundy, Stephen\"},{\"Person.name\":\"González-Losada, Pedro\"},{\"Person.name\":\"Sillankorva, Sanna M.\"}]
datacite.contributors.contributor.contributorName.fl_str_mv RepositóriUM - Universidade do Minho
datacite.creators.creator.creatorName.fl_str_mv Vinayakumar, K. B.
Silva, Maria Daniela
Martins, Artur
Mundy, Stephen
González-Losada, Pedro
Sillankorva, Sanna M.
datacite.date.Accepted.fl_str_mv 2023-06-01T00:00:00Z
datacite.date.available.fl_str_mv 2023-06-20T08:40:40Z
datacite.date.embargoed.fl_str_mv 2023-06-20T08:40:40Z
datacite.rights.fl_str_mv http://purl.org/coar/access_right/c_abf2
datacite.subjects.subject.fl_str_mv 3D printing
biofilms
Klebsiella pneumoniae
levofloxacin
microneedles
polyvinyl alcohol
datacite.titles.title.fl_str_mv Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
dc.contributor.none.fl_str_mv RepositóriUM - Universidade do Minho
dc.creator.none.fl_str_mv Vinayakumar, K. B.
Silva, Maria Daniela
Martins, Artur
Mundy, Stephen
González-Losada, Pedro
Sillankorva, Sanna M.
dc.date.Accepted.fl_str_mv 2023-06-01T00:00:00Z
dc.date.available.fl_str_mv 2023-06-20T08:40:40Z
dc.date.embargoed.fl_str_mv 2023-06-20T08:40:40Z
dc.format.none.fl_str_mv application/pdf
dc.identifier.none.fl_str_mv https://hdl.handle.net/1822/85094
dc.language.none.fl_str_mv eng
dc.publisher.none.fl_str_mv Wiley
dc.rights.none.fl_str_mv http://purl.org/coar/access_right/c_abf2
dc.subject.none.fl_str_mv 3D printing
biofilms
Klebsiella pneumoniae
levofloxacin
microneedles
polyvinyl alcohol
dc.title.fl_str_mv Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
dc.type.none.fl_str_mv http://purl.org/coar/resource_type/c_6501
description Additive manufacturing advancements contribute considerably to several fields, and its use in the medical field is gaining attention due to its easily customizable option (patient-specific), low cost, and fast turnout time in developing drug delivery and diagnostic tools. Here, wereport the fabrication of a microneedle (MN) platform using a stereolithography 3D printer, varying the 3D printing angle and aspect ratio (2:1, 3:1, 4:1). The optimal printing angle was30, resulting in needle tip and base diameters of 50 µm and 330 µm, and heights of 550/850/1180 µm. Polyvinyl alcohol (PVA) MNs produced with varying levofloxacin concentrations showed variability of 4% in tip and 3% base diameters and 15% in height compared to the 3D-printed MNs. Geometry B wasused to produce levofloxacin-loaded PVA MNs and tested against Klebsiella pneumoniae colony biofilms. Levofloxacin wasreleased gradually, as assessed by spectrofluorimetry. The MIC of levofloxacin against the K. pneumoniae clinical isolate was4 µg/mL, but this concentration wasinsufficient to cause any effect on K. pneumoniae biofilms. Only concentrations 32 µg/mL werestatistically different compared to the unloaded MNs. 3D printing is an attractive solution to produce molds for fabricating biopolymeric MNs for topical drug delivery.
dirty 0
eu_rights_str_mv openAccess
format article
fulltext.url.fl_str_mv https://repositorium.uminho.pt/bitstreams/3ff9b921-0049-4476-8a21-9fb7116a4647/download
id rum_8ec1e2d27fdc2f747e744c094e0825a3
identifier.url.fl_str_mv https://hdl.handle.net/1822/85094
instacron_str repositorium
institution Universidade do Minho
instname_str Universidade do Minho
language eng
network_acronym_str rum
network_name_str RepositóriUM - Universidade do Minho
oai_identifier_str oai:repositorium.uminho.pt:1822/85094
organization_str_mv urn:organizationAcronym:repositorium
person_str_mv Vinayakumar, K. B.
Silva, Maria Daniela
Martins, Artur
Mundy, Stephen
González-Losada, Pedro
Sillankorva, Sanna M.
publishDate 2023
publisher.none.fl_str_mv Wiley
reponame_str RepositóriUM - Universidade do Minho
repository_id_str urn:repositoryAcronym:rum
service_str_mv urn:repositoryAcronym:rum
spelling engWileyporAdditive manufacturing advancements contribute considerably to several fields, and its use in the medical field is gaining attention due to its easily customizable option (patient-specific), low cost, and fast turnout time in developing drug delivery and diagnostic tools. Here, wereport the fabrication of a microneedle (MN) platform using a stereolithography 3D printer, varying the 3D printing angle and aspect ratio (2:1, 3:1, 4:1). The optimal printing angle was30, resulting in needle tip and base diameters of 50 µm and 330 µm, and heights of 550/850/1180 µm. Polyvinyl alcohol (PVA) MNs produced with varying levofloxacin concentrations showed variability of 4% in tip and 3% base diameters and 15% in height compared to the 3D-printed MNs. Geometry B wasused to produce levofloxacin-loaded PVA MNs and tested against Klebsiella pneumoniae colony biofilms. Levofloxacin wasreleased gradually, as assessed by spectrofluorimetry. The MIC of levofloxacin against the K. pneumoniae clinical isolate was4 µg/mL, but this concentration wasinsufficient to cause any effect on K. pneumoniae biofilms. Only concentrations 32 µg/mL werestatistically different compared to the unloaded MNs. 3D printing is an attractive solution to produce molds for fabricating biopolymeric MNs for topical drug delivery.application/pdfporLevofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm controlVinayakumar, K. B.Silva, Maria DanielaMartins, ArturMundy, StephenGonzález-Losada, PedroSillankorva, Sanna M.HostingInstitutionOrganizationalRepositóriUM - Universidade do Minhoe-mailmailto:repositorium@usdb.uminho.ptrepositorium@usdb.uminho.ptCITATIONVinayakumar, K. B.; Silva, Maria Daniela; Martins, Artur; Mundy, Stephen; González-Losada, Pedro; Sillankorva, Sanna M., Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control. Advanced Therapeutics, 6(6), 2200320, 2023ISSNIsPartOf2366-3987DOIIsPartOf10.1002/adtp.2022003202023-06-20T08:40:40Z2023-062023-06-17T09:08:07Z2023-06-01T00:00:00ZHandlehttps://hdl.handle.net/1822/85094http://purl.org/coar/access_right/c_abf2open access3D printingbiofilmsKlebsiella pneumoniaelevofloxacinmicroneedlespolyvinyl alcohol3014501 bytesliteraturehttp://purl.org/coar/resource_type/c_6501journal articlehttp://purl.org/coar/access_right/c_abf2application/pdffulltexthttps://repositorium.uminho.pt/bitstreams/3ff9b921-0049-4476-8a21-9fb7116a4647/download
spellingShingle Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
Vinayakumar, K. B.
3D printing
biofilms
Klebsiella pneumoniae
levofloxacin
microneedles
polyvinyl alcohol
status SINGLETON
subject.fl_str_mv 3D printing
biofilms
Klebsiella pneumoniae
levofloxacin
microneedles
polyvinyl alcohol
title Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
title_full Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
title_fullStr Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
title_full_unstemmed Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
title_short Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
title_sort Levofloxacin-loaded microneedles produced using 3D-printed molds for Klebsiella pneumoniae biofilm control
topic 3D printing
biofilms
Klebsiella pneumoniae
levofloxacin
microneedles
polyvinyl alcohol
topic_facet 3D printing
biofilms
Klebsiella pneumoniae
levofloxacin
microneedles
polyvinyl alcohol
url https://hdl.handle.net/1822/85094
visible 1