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Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides

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Resumo:Maleimides were combined with D-erythrose benzylidene-acetal 1,3-butadienes 1 and 2 to study the facial selectivity of the Diels-Alder cycloadditions. The selectivity was found to be from moderate to good. The reaction diastereotopicity can be reversed with the temperature. Simultaneous coordination of diene 1, having a free hydroxyl group, and maleimide 3 to a chiral bimetallic Lewis acid catalyst (LACASA-DA reaction) occurs with complete diastereo-control to give a single adduct, using an extra chiral inductor either R- or S-BINOL.
Autores principais:Salgueiro, D. A. L.
Outros Autores:Duarte, Vera C. M.; Sousa, Cristina; Alves, M. José; Fortes, A. Gil
Assunto:maleimides D-erythrose benzylidene-acetal 1,3-butadiene Diels-Alder cycloaddition selectivity
Ano:2012
País:Portugal
Tipo de documento:artigo
Tipo de acesso:acesso aberto
Instituição associada:Universidade do Minho
Idioma:inglês
Origem:RepositóriUM - Universidade do Minho
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author Salgueiro, D. A. L.
author2 Duarte, Vera C. M.
Sousa, Cristina
Alves, M. José
Fortes, A. Gil
author2_role author
author
author
author
author_facet Salgueiro, D. A. L.
Duarte, Vera C. M.
Sousa, Cristina
Alves, M. José
Fortes, A. Gil
author_role author
contributor_name_str_mv RepositóriUM - Universidade do Minho
country_str PT
creators_json_txt [{\"Person.name\":\"Salgueiro, D. A. L.\"},{\"Person.name\":\"Duarte, Vera C. M.\"},{\"Person.name\":\"Sousa, Cristina\"},{\"Person.name\":\"Alves, M. José\"},{\"Person.name\":\"Fortes, A. Gil\"}]
datacite.contributors.contributor.contributorName.fl_str_mv RepositóriUM - Universidade do Minho
datacite.creators.creator.creatorName.fl_str_mv Salgueiro, D. A. L.
Duarte, Vera C. M.
Sousa, Cristina
Alves, M. José
Fortes, A. Gil
datacite.date.Accepted.fl_str_mv 2012-01-01T00:00:00Z
datacite.date.available.fl_str_mv 2012-12-21T18:24:28Z
datacite.date.embargoed.fl_str_mv 2012-12-21T18:24:28Z
datacite.rights.fl_str_mv http://purl.org/coar/access_right/c_abf2
datacite.subjects.subject.fl_str_mv maleimides
D-erythrose benzylidene-acetal 1,3-butadiene
Diels-Alder cycloaddition
selectivity
datacite.titles.title.fl_str_mv Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
dc.contributor.none.fl_str_mv RepositóriUM - Universidade do Minho
dc.creator.none.fl_str_mv Salgueiro, D. A. L.
Duarte, Vera C. M.
Sousa, Cristina
Alves, M. José
Fortes, A. Gil
dc.date.Accepted.fl_str_mv 2012-01-01T00:00:00Z
dc.date.available.fl_str_mv 2012-12-21T18:24:28Z
dc.date.embargoed.fl_str_mv 2012-12-21T18:24:28Z
dc.format.none.fl_str_mv application/pdf
dc.identifier.none.fl_str_mv https://hdl.handle.net/1822/22057
dc.language.none.fl_str_mv eng
dc.publisher.none.fl_str_mv Georg Thieme Verlag
dc.rights.none.fl_str_mv http://purl.org/coar/access_right/c_abf2
dc.subject.none.fl_str_mv maleimides
D-erythrose benzylidene-acetal 1,3-butadiene
Diels-Alder cycloaddition
selectivity
dc.title.fl_str_mv Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
dc.type.none.fl_str_mv http://purl.org/coar/resource_type/c_6501
description Maleimides were combined with D-erythrose benzylidene-acetal 1,3-butadienes 1 and 2 to study the facial selectivity of the Diels-Alder cycloadditions. The selectivity was found to be from moderate to good. The reaction diastereotopicity can be reversed with the temperature. Simultaneous coordination of diene 1, having a free hydroxyl group, and maleimide 3 to a chiral bimetallic Lewis acid catalyst (LACASA-DA reaction) occurs with complete diastereo-control to give a single adduct, using an extra chiral inductor either R- or S-BINOL.
dirty 0
eu_rights_str_mv openAccess
format article
fulltext.url.fl_str_mv https://repositorium.uminho.pt/bitstreams/35e62a9b-523a-48d1-bec6-11953b70ee93/download
id rum_1dafe00601df96feff436c0e082c2f71
identifier.url.fl_str_mv https://hdl.handle.net/1822/22057
instacron_str repositorium
institution Universidade do Minho
instname_str Universidade do Minho
language eng
network_acronym_str rum
network_name_str RepositóriUM - Universidade do Minho
oai_identifier_str oai:repositorium.uminho.pt:1822/22057
organization_str_mv urn:organizationAcronym:repositorium
person_str_mv Salgueiro, D. A. L.
Duarte, Vera C. M.
Sousa, Cristina
Alves, M. José
Fortes, A. Gil
publishDate 2012
publisher.none.fl_str_mv Georg Thieme Verlag
reponame_str RepositóriUM - Universidade do Minho
repository_id_str urn:repositoryAcronym:rum
service_str_mv urn:repositoryAcronym:rum
spelling engGeorg Thieme VerlagMaleimides were combined with D-erythrose benzylidene-acetal 1,3-butadienes 1 and 2 to study the facial selectivity of the Diels-Alder cycloadditions. The selectivity was found to be from moderate to good. The reaction diastereotopicity can be reversed with the temperature. Simultaneous coordination of diene 1, having a free hydroxyl group, and maleimide 3 to a chiral bimetallic Lewis acid catalyst (LACASA-DA reaction) occurs with complete diastereo-control to give a single adduct, using an extra chiral inductor either R- or S-BINOL.application/pdfporDiastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimidesSalgueiro, D. A. L.Duarte, Vera C. M.Sousa, CristinaAlves, M. JoséFortes, A. GilHostingInstitutionOrganizationalRepositóriUM - Universidade do Minhoe-mailmailto:repositorium@usdb.uminho.ptrepositorium@usdb.uminho.ptISSNIsPartOf0936-5214DOIIsPartOf10.1055/s-0031-12897852012-12-21T18:24:28Z20122012-01-01T00:00:00ZHandlehttps://hdl.handle.net/1822/22057http://purl.org/coar/access_right/c_abf2open accessmaleimidesD-erythrose benzylidene-acetal 1,3-butadieneDiels-Alder cycloadditionselectivity331330 bytesliteraturehttp://purl.org/coar/resource_type/c_6501journal articlehttp://purl.org/coar/access_right/c_abf2application/pdffulltexthttps://repositorium.uminho.pt/bitstreams/35e62a9b-523a-48d1-bec6-11953b70ee93/download
spellingShingle Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
Salgueiro, D. A. L.
maleimides
D-erythrose benzylidene-acetal 1,3-butadiene
Diels-Alder cycloaddition
selectivity
status SINGLETON
subject.fl_str_mv maleimides
D-erythrose benzylidene-acetal 1,3-butadiene
Diels-Alder cycloaddition
selectivity
title Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
title_full Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
title_fullStr Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
title_full_unstemmed Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
title_short Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
title_sort Diastereo-selectivity in diels–alder cycloadditions of erythrose benzylidene-acetal 1,3-Butadienes with maleimides
topic maleimides
D-erythrose benzylidene-acetal 1,3-butadiene
Diels-Alder cycloaddition
selectivity
topic_facet maleimides
D-erythrose benzylidene-acetal 1,3-butadiene
Diels-Alder cycloaddition
selectivity
url https://hdl.handle.net/1822/22057
visible 1