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Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody

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Resumo:Monoclonal antibody-based therapy has shown efficacy against cancer, autoimmune, infectious, and inflammatory diseases. Multispecific antibodies (MsAbs), including trispecifics (tsAbs), offer enhanced therapeutic potential by targeting different epitopes. However, when co-expressed from three or more different polypeptide chains, MsAb production can lead to incorrect chain assembly and co-production of mispaired species with impaired biological activity. Moreover, mispairing carries significant challenges for downstream purification, decreasing yields and increasing the cost of bioprocess development. In this study, quantitative transcriptomics and proteomics analyses were employed to investigate which signaling pathways correlated with low and high mispairing clone signatures. Gene and protein expression profiles of Chinese hamster ovary (CHO) clones producing an tsAb were analyzed in the exponential growth and stationary (tsAb production) phase of fed-batch culture. Functional analysis revealed activated endoplasmic reticulum stress in high mispairing clones in both culture phases, while low mispairing clones exhibited expression profiles indicative of activated protein translation, as well as higher endocytosis and target protein degradation, suggesting the clearance of unfolded proteins through ubiquitin-mediated mechanisms. In addition, through transcriptomic profiling, we identified a group of genes that have the potential to be used as a biomarker panel tool for identifying high mispairing levels in the early stages of bioprocess development.
Autores principais:Sebastião, Maria João
Outros Autores:Hoffman, Michael; Escandell, José; Tousi, Fatemeh; Zhang, Jin; Figueroa, Bruno; DeMaria, Christine; Gomes-Alves, Patrícia
Assunto:CHO cells mispairing multispecific antibodies proteomics transcriptomics Medicine (miscellaneous) General Biochemistry,Genetics and Molecular Biology SDG 3 - Good Health and Well-being
Ano:2023
País:Portugal
Tipo de documento:artigo
Tipo de acesso:acesso aberto
Instituição associada:Universidade Nova de Lisboa
Idioma:inglês
Origem:Repositório Institucional da UNL
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author Sebastião, Maria João
author2 Hoffman, Michael
Escandell, José
Tousi, Fatemeh
Zhang, Jin
Figueroa, Bruno
DeMaria, Christine
Gomes-Alves, Patrícia
author2_role author
author
author
author
author
author
author
author_facet Sebastião, Maria João
Hoffman, Michael
Escandell, José
Tousi, Fatemeh
Zhang, Jin
Figueroa, Bruno
DeMaria, Christine
Gomes-Alves, Patrícia
author_role author
contributor_name_str_mv Instituto de Tecnologia Química e Biológica António Xavier (ITQB)
MDPI AG
RUN
country_str PT
creators_json_txt [{\"Person.name\":\"Sebastião, Maria João\"},{\"Person.name\":\"Hoffman, Michael\"},{\"Person.name\":\"Escandell, José\"},{\"Person.name\":\"Tousi, Fatemeh\"},{\"Person.name\":\"Zhang, Jin\"},{\"Person.name\":\"Figueroa, Bruno\"},{\"Person.name\":\"DeMaria, Christine\"},{\"Person.name\":\"Gomes-Alves, Patrícia\"}]
datacite.contributors.contributor.contributorName.fl_str_mv Instituto de Tecnologia Química e Biológica António Xavier (ITQB)
MDPI AG
RUN
datacite.creators.creator.creatorName.fl_str_mv Sebastião, Maria João
Hoffman, Michael
Escandell, José
Tousi, Fatemeh
Zhang, Jin
Figueroa, Bruno
DeMaria, Christine
Gomes-Alves, Patrícia
datacite.date.Accepted.fl_str_mv 2023-11-01T00:00:00Z
datacite.date.available.fl_str_mv 2024-04-02T23:52:23Z
datacite.date.embargoed.fl_str_mv 2024-04-02T23:52:23Z
datacite.rights.fl_str_mv http://purl.org/coar/access_right/c_abf2
datacite.subjects.subject.fl_str_mv CHO cells
mispairing
multispecific antibodies
proteomics
transcriptomics
Medicine (miscellaneous)
General Biochemistry,Genetics and Molecular Biology
SDG 3 - Good Health and Well-being
datacite.titles.title.fl_str_mv Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
dc.contributor.none.fl_str_mv Instituto de Tecnologia Química e Biológica António Xavier (ITQB)
MDPI AG
RUN
dc.creator.none.fl_str_mv Sebastião, Maria João
Hoffman, Michael
Escandell, José
Tousi, Fatemeh
Zhang, Jin
Figueroa, Bruno
DeMaria, Christine
Gomes-Alves, Patrícia
dc.date.Accepted.fl_str_mv 2023-11-01T00:00:00Z
dc.date.available.fl_str_mv 2024-04-02T23:52:23Z
dc.date.embargoed.fl_str_mv 2024-04-02T23:52:23Z
dc.format.none.fl_str_mv application/pdf
dc.identifier.none.fl_str_mv http://hdl.handle.net/10362/165743
dc.language.none.fl_str_mv eng
dc.rights.none.fl_str_mv http://purl.org/coar/access_right/c_abf2
dc.subject.none.fl_str_mv CHO cells
mispairing
multispecific antibodies
proteomics
transcriptomics
Medicine (miscellaneous)
General Biochemistry,Genetics and Molecular Biology
SDG 3 - Good Health and Well-being
dc.title.fl_str_mv Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
dc.type.none.fl_str_mv http://purl.org/coar/resource_type/c_6501
description Monoclonal antibody-based therapy has shown efficacy against cancer, autoimmune, infectious, and inflammatory diseases. Multispecific antibodies (MsAbs), including trispecifics (tsAbs), offer enhanced therapeutic potential by targeting different epitopes. However, when co-expressed from three or more different polypeptide chains, MsAb production can lead to incorrect chain assembly and co-production of mispaired species with impaired biological activity. Moreover, mispairing carries significant challenges for downstream purification, decreasing yields and increasing the cost of bioprocess development. In this study, quantitative transcriptomics and proteomics analyses were employed to investigate which signaling pathways correlated with low and high mispairing clone signatures. Gene and protein expression profiles of Chinese hamster ovary (CHO) clones producing an tsAb were analyzed in the exponential growth and stationary (tsAb production) phase of fed-batch culture. Functional analysis revealed activated endoplasmic reticulum stress in high mispairing clones in both culture phases, while low mispairing clones exhibited expression profiles indicative of activated protein translation, as well as higher endocytosis and target protein degradation, suggesting the clearance of unfolded proteins through ubiquitin-mediated mechanisms. In addition, through transcriptomic profiling, we identified a group of genes that have the potential to be used as a biomarker panel tool for identifying high mispairing levels in the early stages of bioprocess development.
dirty 0
eu_rights_str_mv openAccess
format article
fulltext.url.fl_str_mv https://run.unl.pt/bitstreams/a892e93f-9ee4-43b0-b9fb-98055396159c/download
id run_ac2bef3cbafc8dc1e44019a5f596fb34
identifier.url.fl_str_mv http://hdl.handle.net/10362/165743
inst_facet_str urn:organizationAcronym:unl{{{_:::_}}}Universidade Nova de Lisboa
instacron_str unl
institution Universidade Nova de Lisboa
instname_str Universidade Nova de Lisboa
language eng
network_acronym_str run
network_name_str Repositório Institucional da UNL
oai_identifier_str oai:run.unl.pt:10362/165743
organization_str_mv urn:organizationAcronym:unl
person_str_mv Sebastião, Maria João
Hoffman, Michael
Escandell, José
Tousi, Fatemeh
Zhang, Jin
Figueroa, Bruno
DeMaria, Christine
Gomes-Alves, Patrícia
publishDate 2023
repo_facet_str urn:repositoryAcronym:run{{{_:::_}}}Repositório Institucional da UNL
reponame_str Repositório Institucional da UNL
repository_id_str urn:repositoryAcronym:run
service_str_mv urn:repositoryAcronym:run
spelling engenMonoclonal antibody-based therapy has shown efficacy against cancer, autoimmune, infectious, and inflammatory diseases. Multispecific antibodies (MsAbs), including trispecifics (tsAbs), offer enhanced therapeutic potential by targeting different epitopes. However, when co-expressed from three or more different polypeptide chains, MsAb production can lead to incorrect chain assembly and co-production of mispaired species with impaired biological activity. Moreover, mispairing carries significant challenges for downstream purification, decreasing yields and increasing the cost of bioprocess development. In this study, quantitative transcriptomics and proteomics analyses were employed to investigate which signaling pathways correlated with low and high mispairing clone signatures. Gene and protein expression profiles of Chinese hamster ovary (CHO) clones producing an tsAb were analyzed in the exponential growth and stationary (tsAb production) phase of fed-batch culture. Functional analysis revealed activated endoplasmic reticulum stress in high mispairing clones in both culture phases, while low mispairing clones exhibited expression profiles indicative of activated protein translation, as well as higher endocytosis and target protein degradation, suggesting the clearance of unfolded proteins through ubiquitin-mediated mechanisms. In addition, through transcriptomic profiling, we identified a group of genes that have the potential to be used as a biomarker panel tool for identifying high mispairing levels in the early stages of bioprocess development.application/pdfenIdentification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific AntibodySebastião, Maria JoãoHoffman, MichaelEscandell, JoséTousi, FatemehZhang, JinFigueroa, BrunoDeMaria, ChristineGomes-Alves, PatríciaInstituto de Tecnologia Química e Biológica António Xavier (ITQB)MDPI AGHostingInstitutionOrganizationalRUNe-mailmailto:run@unl.ptrun@unl.ptISSNIsPartOf2227-9059URNIsPartOfPURE: 83729506URNIsPartOfPURE UUID: 7e7c218b-2d4c-49f1-be10-2f32f14a083cURNIsPartOfScopus: 85178360671DOIIsPartOf10.3390/biomedicines111128902024-04-02T23:52:23Z2023-112023-11-01T00:00:00ZHandlehttp://hdl.handle.net/10362/165743http://purl.org/coar/access_right/c_abf2open accessCHO cellsmispairingmultispecific antibodiesproteomicstranscriptomicsMedicine (miscellaneous)General Biochemistry,Genetics and Molecular BiologySDG 3 - Good Health and Well-being3081595 bytesliteraturehttp://purl.org/coar/resource_type/c_6501journal articlehttp://purl.org/coar/access_right/c_abf2application/pdffulltexthttps://run.unl.pt/bitstreams/a892e93f-9ee4-43b0-b9fb-98055396159c/download
spellingShingle Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
Sebastião, Maria João
CHO cells
mispairing
multispecific antibodies
proteomics
transcriptomics
Medicine (miscellaneous)
General Biochemistry,Genetics and Molecular Biology
SDG 3 - Good Health and Well-being
status SINGLETON
subject.fl_str_mv CHO cells
mispairing
multispecific antibodies
proteomics
transcriptomics
Medicine (miscellaneous)
General Biochemistry,Genetics and Molecular Biology
SDG 3 - Good Health and Well-being
title Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
title_full Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
title_fullStr Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
title_full_unstemmed Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
title_short Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
title_sort Identification of Mispairing Omic Signatures in Chinese Hamster Ovary (CHO) Cells Producing a Tri-Specific Antibody
topic CHO cells
mispairing
multispecific antibodies
proteomics
transcriptomics
Medicine (miscellaneous)
General Biochemistry,Genetics and Molecular Biology
SDG 3 - Good Health and Well-being
topic_facet CHO cells
mispairing
multispecific antibodies
proteomics
transcriptomics
Medicine (miscellaneous)
General Biochemistry,Genetics and Molecular Biology
SDG 3 - Good Health and Well-being
url http://hdl.handle.net/10362/165743
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